ALBERT — All Library Books, journals and Electronic Records Telegrafenberg

1

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Discovery of a Bicyclic Peptidyl Pan-Ras Inhibitor (2021)

Buyanova, Marina ; Cai, Shurui ; Cooper, Jahan ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c01130. Published 2021 Aug 20. doi: 10.1021/acs.jmedchem.1c01130. [early online release]

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Publication Date: 2021-08-20

Print ISSN: 0022-2623

Electronic ISSN: 1520-4804

Topics: Chemistry and Pharmacology , Medicine

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2

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Mechanistic Investigation of Site-specific DNA Methylating Agents Targeting Breast Cancer Cells (2021)

Lowder, Leah L. ; Powell, Matthew ; Miller, Sean E. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c00615. Published 2021 Aug 20. doi: 10.1021/acs.jmedchem.1c00615. [early online release]

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Publication Date: 2021-08-20

Print ISSN: 0022-2623

Electronic ISSN: 1520-4804

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3

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Interrogating the Inhibition Mechanisms of Human Aldehyde Oxidase by X-ray Crystallography and NMR Spectroscopy: The Raloxifene Case (2021)

Mota, Cristiano ; Diniz, Ana ; Coelho, Catarina ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c01125. Published 2021 Aug 20. doi: 10.1021/acs.jmedchem.1c01125. [early online release]

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Publication Date: 2021-08-20

Print ISSN: 0022-2623

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Published by American Chemical Society

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4

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1,3-Diarylpyrazolyl-acylsulfonamides as Potent Anti-tuberculosis Agents Targeting Cell Wall Biosynthesis in Mycobacterium tuberculosis (2021)

Khonde, Lutete Peguy ; Müller, Rudolf ; Boyle, Grant A. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c00837. Published 2021 Aug 20. doi: 10.1021/acs.jmedchem.1c00837. [early online release]

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Publication Date: 2021-08-20

Print ISSN: 0022-2623

Electronic ISSN: 1520-4804

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Published by American Chemical Society

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5

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Probing the Allosteric Inhibition Mechanism of a Spike Protein Using Molecular Dynamics Simulations and Active Compound Identifications (2021)

Wang, Qian ; Wang, Lin ; Zhang, Yumin ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c00320. Published 2021 Aug 20. doi: 10.1021/acs.jmedchem.1c00320. [early online release]

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Publication Date: 2021-08-20

Print ISSN: 0022-2623

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6

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Pharmacophore-Based Design of Phenyl-[hydroxycyclohexyl] Cycloalkyl-Carboxamide Mitofusin Activators with Improved Neuronal Activity (2021)

Dang, Xiawei ; Williams, Sidney B. ; Devanathan, Sriram ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c00163. Published 2021 Aug 20. doi: 10.1021/acs.jmedchem.1c00163. [early online release]

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Publication Date: 2021-08-20

Print ISSN: 0022-2623

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7

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Discovery of N-(4-(3-isopropyl-2-methyl-2H-indazol-5-yl)pyrimidin-2-yl)-4-(4-methylpiperazin-1-yl)quinazolin-7-amine as a Novel, Potent, and Oral Cyclin-Dependent Kinase Inhibitor against Haematological Malignancies (2021)

Huang, Jianhang ; Wang, Xinren ; Dong, Ruinan ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c00271. Published 2021 Aug 20. doi: 10.1021/acs.jmedchem.1c00271. [early online release]

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Publication Date: 2021-08-20

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8

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Structure-Based Exploration of Selectivity for ATM Inhibitors in Huntington’s Disease (2021)

Van de Poël, Amanda ; Toledo-Sherman, Leticia ; Breccia, Perla ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c00114. Published 2021 Mar 30. doi: 10.1021/acs.jmedchem.1c00114. [early online release]

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Publication Date: 2021-03-30

Print ISSN: 0022-2623

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9

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Direct Observation of Protonation State Modulation in SARS-CoV-2 Main Protease upon Inhibitor Binding with Neutron Crystallography (2021)

Kneller, Daniel W. ; Phillips, Gwyndalyn ; Weiss, Kevin L. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c00058. Published 2021 Mar 23. doi: 10.1021/acs.jmedchem.1c00058. [early online release]

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Publication Date: 2021-03-23

Print ISSN: 0022-2623

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10

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Illuminating a Dark Kinase: Structure-Guided Design, Synthesis, and Evaluation of a Potent Nek1 Inhibitor and Its Effects on the Embryonic Zebrafish Pronephros (2021)

Baumann, Georg ; Meckel, Tobias ; Böhm, Kevin ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.0c02118. Published 2021 Mar 16. doi: 10.1021/acs.jmedchem.0c02118. [early online release]

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Publication Date: 2021-03-16

Print ISSN: 0022-2623

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11

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Remdesivir Metabolite GS-441524 Effectively Inhibits SARS-CoV-2 Infection in Mouse Models (2021)

Li, Yingjun ; Cao, Liu ; Li, Ge ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.0c01929. Published 2021 Feb 01. doi: 10.1021/acs.jmedchem.0c01929. [early online release]

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Publication Date: 2021-02-01

Print ISSN: 0022-2623

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12

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Carboxylesterase Notum Is a Druggable Target to Modulate Wnt Signaling (2021)

Bayle, Elliott D. ; Svensson, Fredrik ; Atkinson, Benjamin N. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.0c01974. Published 2021 Mar 30. doi: 10.1021/acs.jmedchem.0c01974. [early online release]

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Publication Date: 2021-03-30

Print ISSN: 0022-2623

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13

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Discovery of Novel Pyrrolo[2,3-d]pyrimidine-based Derivatives as Potent JAK/HDAC Dual Inhibitors for the Treatment of Refractory Solid Tumors (2021)

Liang, Xuewu ; Tang, Shuai ; Liu, Xuyi ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.0c02111. Published 2021 Feb 15. doi: 10.1021/acs.jmedchem.0c02111. [early online release]

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Publication Date: 2021-02-15

Print ISSN: 0022-2623

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14

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Structural Determinants for the Mode of Action of Imidazopyridine DS2 at δ-Containing γ-Aminobutyric Acid Type A Receptors (2021)

Rostrup, Frederik ; Falk-Petersen, Christina B. ; Harpso̷e, Kasper ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4730-4743. Published 2021 Apr 13. doi: 10.1021/acs.jmedchem.0c02163.

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Publication Date: 2021-04-13

Print ISSN: 0022-2623

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Published by American Chemical Society

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15

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What’s in a Name? Drug Nomenclature and Medicinal Chemistry Trends using INN Publications (2021)

Serafini, Marta ; Cargnin, Sarah ; Massarotti, Alberto ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4410-4429. Published 2021 Apr 13. doi: 10.1021/acs.jmedchem.1c00181.

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Publication Date: 2021-04-13

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16

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First-Time Disclosure of CVN424, a Potent and Selective GPR6 Inverse Agonist for the Treatment of Parkinson’s Disease: Discovery, Pharmacological Validation, and Identification of a Clinical Candidate (2021)

Sun, Huikai ; Monenschein, Holger ; Schiffer, Hans H. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.0c02081. Published 2021 Apr 16. doi: 10.1021/acs.jmedchem.0c02081. [early online release]

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Publication Date: 2021-04-16

Print ISSN: 0022-2623

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Topics: Chemistry and Pharmacology , Medicine

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17

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Antimicrobial Bombinin-like Peptide 3 Selectively Recognizes and Inserts into Bacterial Biomimetic Bilayers in Multiple Steps (2021)

Annaval, Thibault ; Ramos-Martín, Francisco ; Herrera-León, Claudia ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5185-5197. Published 2021 Apr 14. doi: 10.1021/acs.jmedchem.1c00310.

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Publication Date: 2021-04-14

Print ISSN: 0022-2623

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18

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Tetrahydroquinoline-Capped Histone Deacetylase 6 Inhibitor SW-101 Ameliorates Pathological Phenotypes in a Charcot–Marie–Tooth Type 2A Mouse Model (2021)

Shen, Sida ; Picci, Cristina ; Ustinova, Kseniya ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4810-4840. Published 2021 Apr 08. doi: 10.1021/acs.jmedchem.0c02210.

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Publication Date: 2021-04-08

Print ISSN: 0022-2623

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19

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GPR120/FFAR4 Pharmacology: Focus on Agonists in Type 2 Diabetes Mellitus Drug Discovery (2021)

Carullo, Gabriele ; Mazzotta, Sarah ; Vega-Holm, Margarita ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4312-4332. Published 2021 Apr 10. doi: 10.1021/acs.jmedchem.0c01002.

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Publication Date: 2021-04-10

Print ISSN: 0022-2623

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20

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Sustainable Drug Discovery of Multi-Target-Directed Ligands for Alzheimer’s Disease (2021)

Rossi, Michele ; Freschi, Michela ; de Camargo Nascente, Luciana ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4972-4990. Published 2021 Apr 08. doi: 10.1021/acs.jmedchem.1c00048.

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Publication Date: 2021-04-08

Print ISSN: 0022-2623

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21

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Antimalarial Benzimidazole Derivatives Incorporating Phenolic Mannich Base Side Chains Inhibit Microtubule and Hemozoin Formation: Structure–Activity Relationship and In Vivo Oral Efficacy Studies (2021)

Dziwornu, Godwin Akpeko ; Coertzen, Dina ; Leshabane, Meta ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5198-5215. Published 2021 Apr 12. doi: 10.1021/acs.jmedchem.1c00354.

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Publication Date: 2021-04-12

Print ISSN: 0022-2623

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22

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Correction to Assessment of NR4A Ligands That Directly Bind and Modulate the Orphan Nuclear Receptor Nurr1 (2021)

Munoz-Tello, Paola ; Lin, Hua ; Khan, Pasha ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5216-5220. Published 2021 Apr 12. doi: 10.1021/acs.jmedchem.1c00526.

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Publication Date: 2021-04-12

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23

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Tuberculosis: An Overview of the Immunogenic Response, Disease Progression, and Medicinal Chemistry Efforts in the Last Decade toward the Development of Potential Drugs for Extensively Drug-Resistant Tuberculosis Strains (2021)

Sharma, Akanksha ; De Rosa, Maria ; Singla, Neha ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4359-4395. Published 2021 Apr 07. doi: 10.1021/acs.jmedchem.0c01833.

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Publication Date: 2021-04-07

Print ISSN: 0022-2623

Electronic ISSN: 1520-4804

Topics: Chemistry and Pharmacology , Medicine

Published by American Chemical Society

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24

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Tricyclic Triazoles as σ1 Receptor Antagonists for Treating Pain (2021)

Díaz, José Luis ; Cuevas, Félix ; Oliva, Ana I. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5157-5170. Published 2021 Apr 07. doi: 10.1021/acs.jmedchem.1c00244.

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Publication Date: 2021-04-07

Print ISSN: 0022-2623

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25

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Insights into SARS-CoV-2’s Mutations for Evading Human Antibodies: Sacrifice and Survival (2021)

Luan, Binquan ; Huynh, Tien

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c00311. Published 2021 Apr 09. doi: 10.1021/acs.jmedchem.1c00311. [early online release]

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Publication Date: 2021-04-09

Print ISSN: 0022-2623

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26

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Exendin 4-Hapten Conjugate Capable of Binding with Endogenous Antibodies for Peptide Half-life Extension and Exerting Long-Acting Hypoglycemic Activity (2021)

Dai, Shijie ; Hong, Haofei ; Zhou, Kun ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4947-4959. Published 2021 Apr 07. doi: 10.1021/acs.jmedchem.1c00032.

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Publication Date: 2021-04-07

Print ISSN: 0022-2623

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27

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Prodrugs of a 1′-CN-4-Aza-7,9-dideazaadenosine C-Nucleoside Leading to the Discovery of Remdesivir (GS-5734) as a Potent Inhibitor of Respiratory Syncytial Virus with Efficacy in the African Green Monkey Model of RSV (2021)

Mackman, Richard L. ; Hui, Hon C. ; Perron, Michel ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5001-5017. Published 2021 Apr 09. doi: 10.1021/acs.jmedchem.1c00071.

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Publication Date: 2021-04-09

Print ISSN: 0022-2623

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28

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Synthesis of the Potent, Selective, and Efficacious β-Secretase (BACE1) Inhibitor NB-360 (2021)

Rueeger, Heinrich ; Lueoend, Rainer ; Machauer, Rainer ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4677-4696. Published 2021 Apr 12. doi: 10.1021/acs.jmedchem.0c02143.

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Publication Date: 2021-04-12

Print ISSN: 0022-2623

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29

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Three-Dimensional Proteome-Wide Scale Screening for the 5-Alpha Reductase Inhibitor Finasteride: Identification of a Novel Off-Target (2021)

Giatti, Silvia ; Di Domizio, Alessandro ; Diviccaro, Silvia ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4553-4566. Published 2021 Apr 12. doi: 10.1021/acs.jmedchem.0c02039.

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Publication Date: 2021-04-12

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30

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Discovery of AG-270, a First-in-Class Oral MAT2A Inhibitor for the Treatment of Tumors with Homozygous MTAP Deletion (2021)

Konteatis, Zenon ; Travins, Jeremy ; Gross, Stefan ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4430-4449. Published 2021 Apr 08. doi: 10.1021/acs.jmedchem.0c01895.

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Publication Date: 2021-04-08

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31

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A New Turn in Peptide-Based Imaging Agents: Foldamers Afford Improved Theranostics Targeting Cholecystokinin-2 Receptor-Positive Cancer (2021)

Corlett, Alicia ; Sani, Marc-Antoine ; Van Zuylekom, Jessica ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4841-4856. Published 2021 Apr 07. doi: 10.1021/acs.jmedchem.0c02213.

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Publication Date: 2021-04-07

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32

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Discovery of 5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine Derivatives as Highly Selective CK2 Inhibitors with Potent Cancer Cell Stemness Inhibition (2021)

Wang, Yuanjiang ; Lv, Zhaodan ; Chen, Feihong ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5082-5098. Published 2021 Apr 09. doi: 10.1021/acs.jmedchem.1c00131.

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Publication Date: 2021-04-09

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33

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Bispecific Estrogen Receptor α Degraders Incorporating Novel Binders Identified Using DNA-Encoded Chemical Library Screening (2021)

Disch, Jeremy S. ; Duffy, Jennifer M. ; Lee, Esther C. Y. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5049-5066. Published 2021 Apr 12. doi: 10.1021/acs.jmedchem.1c00127.

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Publication Date: 2021-04-12

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34

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Progress toward B-Cell Lymphoma 6 BTB Domain Inhibitors for the Treatment of Diffuse Large B-Cell Lymphoma and Beyond (2021)

Ai, Yong ; Hwang, Lucia ; MacKerell, Alexander D. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4333-4358. Published 2021 Apr 12. doi: 10.1021/acs.jmedchem.0c01686.

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Publication Date: 2021-04-12

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35

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Identification of 2,2-Dimethylbutanoic Acid (HST5040), a Clinical Development Candidate for the Treatment of Propionic Acidemia and Methylmalonic Acidemia (2021)

Armstrong, Allison J. ; Henke, Brad R. ; Collado, Maria Sol ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5037-5048. Published 2021 Apr 13. doi: 10.1021/acs.jmedchem.1c00124.

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Publication Date: 2021-04-13

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36

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Hydrophobic Pocket Occupation Design of Difluoro-Biphenyl-Diarylpyrimidines as Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitors: from N-Alkylation to Methyl Hopping on the Pyrimidine Ring (2021)

Ding, Li ; Pannecouque, Christophe ; De Clercq, Erik ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5067-5081. Published 2021 Apr 14. doi: 10.1021/acs.jmedchem.1c00128.

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Interface-Mediated Mechanism of Action—The Root of the Cytoprotective Effect of Immediate-Release Omeprazole (2021)

Lopes-de-Campos, Daniela ; Pereira-Leite, Catarina ; Fontaine, Philippe ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5171-5184. Published 2021 Apr 13. doi: 10.1021/acs.jmedchem.1c00251.

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38

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Beyond Basicity: Discovery of Nonbasic DENV-2 Protease Inhibitors with Potent Activity in Cell Culture (2021)

Kühl, Nikos ; Leuthold, Mila M. ; Behnam, Mira A. M. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.0c02042. Published 2021 Apr 14. doi: 10.1021/acs.jmedchem.0c02042. [early online release]

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39

Unknown

Issue Publication Information (2021)

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): jmv064i008_1473292. Published 2021 Apr 22. doi: 10.1021/jmv064i008_1473292.

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Recent Developments in the Use of Kinase Inhibitors for Management of Viral Infections (2021)

Raghuvanshi, Rinky ; Bharate, Sandip B.

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.0c01467. Published 2021 Feb 04. doi: 10.1021/acs.jmedchem.0c01467. [early online release]

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41

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Design, Synthesis, and Biological Evaluation of Peptidomimetic Aldehydes as Broad-Spectrum Inhibitors against Enterovirus and SARS-CoV-2 (2021)

Dai, Wenhao ; Jochmans, Dirk ; Xie, Hang ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.0c02258. Published 2021 Apr 19. doi: 10.1021/acs.jmedchem.0c02258. [early online release]

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42

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Identification, Characterization, and Suppression of Side Products Formed during the Synthesis of [177Lu]Lu-PSMA-617 (2021)

Martin, Sebastian ; Tönnesmann, Roswitha ; Hierlmeier, Ina ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4960-4971. Published 2021 Apr 07. doi: 10.1021/acs.jmedchem.1c00045.

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43

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Modulation of the H-Bond Basicity of Functional Groups by α-Fluorine-Containing Functions and its Implications for Lipophilicity and Bioisosterism (2021)

Zafrani, Yossi ; Parvari, Galit ; Amir, Dafna ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4516-4531. Published 2021 Apr 12. doi: 10.1021/acs.jmedchem.0c01868.

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44

Unknown

Targeting Chikungunya Virus Replication by Benzoannulene Inhibitors (2021)

Ahmed, S. Kaleem ; Haese, Nicole N. ; Cowan, Jaden T. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4762-4786. Published 2021 Apr 09. doi: 10.1021/acs.jmedchem.0c02183.

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45

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Projected Dose Optimization of Amino- and Hydroxypyrrolidine Purine PI3Kδ Immunomodulators (2021)

Methot, Joey L. ; Zhou, Hua ; McGowan, Meredeth A. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5137-5156. Published 2021 Apr 02. doi: 10.1021/acs.jmedchem.1c00237.

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46

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Mapping Water Thermodynamics on Drug Candidates via Molecular Building Blocks: a Strategy to Improve Ligand Design and Rationalize SAR (2021)

Hüfner-Wulsdorf, Tobias ; Klebe, Gerhard

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4662-4676. Published 2021 Apr 02. doi: 10.1021/acs.jmedchem.0c02115.

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47

Unknown

Issue Editorial Masthead (2021)

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): jmv064i008_1473293. Published 2021 Apr 22. doi: 10.1021/jmv064i008_1473293.

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48

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Discovery of a Potent and Selective FLT3 Inhibitor (Z)-N-(5-((5-Fluoro-2-oxoindolin-3-ylidene)methyl)-4-methyl-1H-pyrrol-3-yl)-3-(pyrrolidin-1-yl)propanamide with Improved Drug-like Properties and Superior Efficacy in FLT3-ITD-Positive Acute Myeloid Leukemia (2021)

Wang, Junwei ; Pan, Xiang ; Song, Yi ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4870-4890. Published 2021 Apr 02. doi: 10.1021/acs.jmedchem.0c02247.

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49

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Polymeric Encapsulation of a Ru(II)-Based Photosensitizer for Folate-Targeted Photodynamic Therapy of Drug Resistant Cancers (2021)

Karges, Johannes ; Tharaud, Mickaël ; Gasser, Gilles

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4612-4622. Published 2021 Apr 05. doi: 10.1021/acs.jmedchem.0c02006.

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50

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Deconstructing Noncovalent Kelch-like ECH-Associated Protein 1 (Keap1) Inhibitors into Fragments to Reconstruct New Potent Compounds (2021)

Pallesen, Jakob S. ; Narayanan, Dilip ; Tran, Kim T. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4623-4661. Published 2021 Apr 05. doi: 10.1021/acs.jmedchem.0c02094.

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51

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Use of Intramolecular 1,5-Sulfur–Oxygen and 1,5-Sulfur–Halogen Interactions in the Design of N-Methyl-5-aryl-N-(2,2,6,6-tetramethylpiperidin-4-yl)-1,3,4-thiadiazol-2-amine SMN2 Splicing Modulators (2021)

Axford, Jake ; Sung, Moo Je ; Manchester, John ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4744-4761. Published 2021 Apr 06. doi: 10.1021/acs.jmedchem.0c02173.

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52

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Targeting Colorectal Cancer with Conjugates of a Glucose Transporter Inhibitor and 5-Fluorouracil (2021)

Chang, Chun-Kai ; Chiu, Pei-Fang ; Yang, Hui-Yi ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4450-4461. Published 2021 Apr 05. doi: 10.1021/acs.jmedchem.0c00897.

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53

Unknown

Optimization of Truncated Glucagon Peptides to Achieve Selective, High Potency, Full Antagonists (2021)

Yang, Bin ; Gelfanov, Vasily M. ; Perez-Tilve, Diego ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4697-4708. Published 2021 Apr 06. doi: 10.1021/acs.jmedchem.0c02069.

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54

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Synthesis and Biological Evaluation of PSMA Ligands with Aromatic Residues and Fluorescent Conjugates Based on Them (2021)

Machulkin, Aleksei E. ; Shafikov, Radik R. ; Uspenskaya, Anastasia A. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4532-4552. Published 2021 Apr 06. doi: 10.1021/acs.jmedchem.0c01935.

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55

Unknown

Structure-Based Design of Selective LONP1 Inhibitors for Probing In Vitro Biology (2021)

Kingsley, Laura J. ; He, Xiaohui ; McNeill, Matthew ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4857-4869. Published 2021 Apr 06. doi: 10.1021/acs.jmedchem.0c02152.

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56

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Structure–Activity Relationship of Heterocyclic P2Y14 Receptor Antagonists: Removal of the Zwitterionic Character with Piperidine Bioisosteres (2021)

Jung, Young-Hwan ; Salmaso, Veronica ; Wen, Zhiwei ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5099-5122. Published 2021 Mar 31. doi: 10.1021/acs.jmedchem.1c00164.

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57

Unknown

Design, Synthesis, and Structural Characterization of Lysine Covalent BH3 Peptides Targeting Mcl-1 (2021)

Gambini, Luca ; Udompholkul, Parima ; Baggio, Carlo ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4903-4912. Published 2021 Apr 02. doi: 10.1021/acs.jmedchem.1c00005.

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58

Unknown

Toward Raman Subcellular Imaging of Endothelial Dysfunction (2021)

Adamczyk, Adriana ; Matuszyk, Ewelina ; Radwan, Basseem ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4396-4409. Published 2021 Apr 06. doi: 10.1021/acs.jmedchem.1c00051.

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59

Unknown

Synthesis and Characterization of the Novel Rodent-Active and CNS-Penetrant P2X7 Receptor Antagonist Lu AF27139 (2021)

Hopper, Allen T. ; Juhl, Martin ; Hornberg, Jorrit ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4891-4902. Published 2021 Apr 06. doi: 10.1021/acs.jmedchem.0c02249.

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60

Unknown

Discovery of Ethyl Ketone-Based Highly Selective HDACs 1, 2, 3 Inhibitors for HIV Latency Reactivation with Minimum Cellular Potency Serum Shift and Reduced hERG Activity (2021)

Yu, Wensheng ; Liu, Jian ; Clausen, Dane ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4709-4729. Published 2021 Apr 02. doi: 10.1021/acs.jmedchem.0c02150.

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61

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Discovery of Novel Benzimidazole and Indazole Analogues as Tubulin Polymerization Inhibitors with Potent Anticancer Activities (2021)

Ren, Yichang ; Wang, Yuxi ; Li, Gang ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4498-4515. Published 2021 Mar 31. doi: 10.1021/acs.jmedchem.0c01837.

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62

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Discovery and Optimization of 2H-1λ2-Pyridin-2-one Inhibitors of Mutant Isocitrate Dehydrogenase 1 for the Treatment of Cancer (2021)

Rohde, Jason M. ; Karavadhi, Surendra ; Pragani, Rajan ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4913-4946. Published 2021 Apr 06. doi: 10.1021/acs.jmedchem.1c00019.

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63

Unknown

Chiral Alkyl Groups at Position 3(1′) of Pyropheophorbide-a Specify Uptake and Retention by Tumor Cells and Are Essential for Effective Photodynamic Therapy (2021)

Cheruku, Ravindra R. ; Tracy, Erin C. ; Tabaczynski, Walter ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4787-4809. Published 2021 Apr 06. doi: 10.1021/acs.jmedchem.0c02090.

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64

Unknown

Small-Molecule Inhibitors Targeting the Canonical WNT Signaling Pathway for the Treatment of Cancer (2021)

Liu, Zhiqing ; Wang, Pingyuan ; Wold, Eric A. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.0c01799. Published 2021 Apr 06. doi: 10.1021/acs.jmedchem.0c01799. [early online release]

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65

Unknown

Structure-Enabled Discovery of Novel Macrocyclic Inhibitors Targeting Glutaminase 1 Allosteric Binding Site (2021)

Xu, Xi ; Wang, Jubo ; Wang, Min ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4588-4611. Published 2021 Apr 01. doi: 10.1021/acs.jmedchem.0c02044.

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66

Unknown

Oxaprozin Analogues as Selective RXR Agonists with Superior Properties and Pharmacokinetics (2021)

Schierle, Simone ; Chaikuad, Apirat ; Lillich, Felix F. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 5123-5136. Published 2021 Apr 01. doi: 10.1021/acs.jmedchem.1c00235.

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67

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From Celecoxib to a Novel Class of Phosphodiesterase 5 Inhibitors: Trisubstituted Pyrazolines as Novel Phosphodiesterase 5 Inhibitors with Extremely High Potency and Phosphodiesterase Isozyme Selectivity (2021)

Abdel-Halim, Mohammad ; Sigler, Sara ; Racheed, Nora A. S. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4462-4477. Published 2021 Apr 01. doi: 10.1021/acs.jmedchem.0c01120.

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68

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Exploring Heteroaromatic Rings as a Replacement for the Labile Amide of Antiplasmodial Pantothenamides (2021)

Guan, Jinming ; Spry, Christina ; Tjhin, Erick T. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(8): 4478-4497. Published 2021 Apr 01. doi: 10.1021/acs.jmedchem.0c01755.

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69

Unknown

Modular Design of Membrane-Active Antibiotics: From Macromolecular Antimicrobials to Small Scorpionlike Peptidomimetics (2021)

Wang, Minghui ; Feng, Xiaoqian ; Gao, Ruixuan ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c00312. Published 2021 Apr 01. doi: 10.1021/acs.jmedchem.1c00312. [early online release]

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70

Unknown

Correction to “Identification of Novel UGT1A1 Variants Including UGT1A1 454C〉A through the Genotyping of Healthy Participants of the HPTN 077 Study” (2021)

Seneviratne, Herana Kamal ; Hamlin, Allyson N. ; Li, Sue ; [et al.]

American Chemical Society

In: ACS Pharmacology . 2021; 4(4): 1462-1462. Published 2021 Jun 29. doi: 10.1021/acsptsci.1c00158.

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Electronic ISSN: 2575-9108

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71

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Issue Publication Information (2021)

American Chemical Society

In: ACS Pharmacology . 2021; 4(4): ptv004i004_1504195. Published 2021 Aug 13. doi: 10.1021/ptv004i004_1504195.

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72

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DNA-Encoded Chemical Libraries: A Comprehensive Review with Succesful Stories and Future Challenges (2021)

Gironda-Martínez, Adrián ; Donckele, Etienne J. ; Samain, Florent ; [et al.]

American Chemical Society

In: ACS Pharmacology . 2021; 4(4): 1265-1279. Published 2021 Jun 14. doi: 10.1021/acsptsci.1c00118.

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73

Unknown

Rosmarinic Acid Potently Detoxifies Amylin Amyloid and Ameliorates Diabetic Pathology in a Transgenic Rat Model of Type 2 Diabetes (2021)

Wu, Ling ; Velander, Paul ; Brown, Anne M. ; [et al.]

American Chemical Society

In: ACS Pharmacology . 2021; 4(4): 1322-1337. Published 2021 Jul 21. doi: 10.1021/acsptsci.1c00028.

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74

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Structure-Based Design of First-Generation Small Molecule Inhibitors Targeting the Catalytic Pockets of AID, APOBEC3A, and APOBEC3B (2021)

King, Justin J. ; Borzooee, Faezeh ; Im, Junbum ; [et al.]

American Chemical Society

In: ACS Pharmacology . 2021; 4(4): 1390-1407. Published 2021 Jul 19. doi: 10.1021/acsptsci.1c00091.

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75

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In Vitro and In Vivo Evaluation of GSK-3 Radioligands in Alzheimer’s Disease: Preliminary Evidence of Sex Differences (2021)

Knight, Ashley C. ; Varlow, Cassis ; Tong, Junchao ; [et al.]

American Chemical Society

In: ACS Pharmacology . 2021; 4(4): 1287-1294. Published 2021 Jul 20. doi: 10.1021/acsptsci.1c00132.

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76

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Pharmacological Inhibition of the Voltage-Gated Sodium Channel NaV1.7 Alleviates Chronic Visceral Pain in a Rodent Model of Irritable Bowel Syndrome (2021)

Jiang, Yan ; Castro, Joel ; Blomster, Linda V. ; [et al.]

American Chemical Society

In: ACS Pharmacology . 2021; 4(4): 1362-1378. Published 2021 Jun 07. doi: 10.1021/acsptsci.1c00072.

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77

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Reconciling Mystical Experiences with Naturalistic Psychedelic Science: Reply to Sanders and Zijlmans (2021)

Jylkkä, Jussi

American Chemical Society

In: ACS Pharmacology . 2021; 4(4): 1468-1470. Published 2021 Jun 08. doi: 10.1021/acsptsci.1c00137.

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78

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Optimization of a Series of 2,3-Dihydrobenzofurans as Highly Potent, Second Bromodomain (BD2)-Selective, Bromo and Extra-Terminal Domain (BET) Inhibitors (2021)

Lucas, Simon C. C. ; Atkinson, Stephen J. ; Chung, Chun-wa ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 10711-10741. Published 2021 Jul 14. doi: 10.1021/acs.jmedchem.1c00344.

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79

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Structure-Guided Design of a “Bump-and-Hole” Bromodomain-Based Degradation Tag (2021)

Nowak, Radosław P. ; Xiong, Yuan ; Kirmani, Nadia ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11637-11650. Published 2021 Jul 19. doi: 10.1021/acs.jmedchem.1c00958.

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80

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Discovery, Structure–Activity Relationships, and In Vivo Evaluation of Novel Aryl Amides as Brain Penetrant Adaptor Protein 2-Associated Kinase 1 (AAK1) Inhibitors for the Treatment of Neuropathic Pain (2021)

Hartz, Richard A ; Ahuja, Vijay T. ; Nara, Susheel J. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11090-11128. Published 2021 Jul 16. doi: 10.1021/acs.jmedchem.1c00472.

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81

Unknown

Discovery of a First-in-Class Inhibitor of the PRMT5–Substrate Adaptor Interaction (2021)

McKinney, David C. ; McMillan, Brian J. ; Ranaghan, Matthew J. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11148-11168. Published 2021 Aug 03. doi: 10.1021/acs.jmedchem.1c00507.

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82

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Optimization of the Urea Linker of Triazolopyridazine MMV665917 Results in a New Anticryptosporidial Lead with Improved Potency and Predicted hERG Safety Margin (2021)

Oboh, Edmund ; Schubert, Tanner J. ; Teixeira, Jose E. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11729-11745. Published 2021 Aug 03. doi: 10.1021/acs.jmedchem.1c01136.

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83

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Fragment-based Scaffold Hopping: Identification of Potent, Selective, and Highly Soluble Bromo and Extra Terminal Domain (BET) Second Bromodomain (BD2) Inhibitors (2021)

Seal, Jonathan T. ; Atkinson, Stephen J. ; Bamborough, Paul ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 10772-10805. Published 2021 Jul 13. doi: 10.1021/acs.jmedchem.1c00365.

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Publication Date: 2021-07-13

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84

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3H-Pyrazolo[4,3-f]quinoline-Based Kinase Inhibitors Inhibit the Proliferation of Acute Myeloid Leukemia Cells In Vivo (2021)

Dayal, Neetu ; Řezníčková, Eva ; Hernandez, Delmis E. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 10981-10996. Published 2021 Jul 21. doi: 10.1021/acs.jmedchem.1c00330.

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85

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Novel Broad-Spectrum Antimicrobial Peptide Derived from Anoplin and Its Activity on Bacterial Pneumonia in Mice (2021)

Gou, Sanhu ; Li, Beibei ; Ouyang, Xu ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11247-11266. Published 2021 Jun 28. doi: 10.1021/acs.jmedchem.1c00614.

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86

Unknown

Discovery and Characterization of Selective and Ligand-Efficient DYRK Inhibitors (2021)

Henderson, Scott H. ; Sorrell, Fiona ; Bennett, James ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11709-11728. Published 2021 Aug 03. doi: 10.1021/acs.jmedchem.1c01115.

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87

Unknown

Current Landscape and Future Perspective of Oxazolidinone Scaffolds Containing Antibacterial Drugs (2021)

Zhao, Qianqian ; Xin, Liang ; Liu, Yuzhi ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 10557-10580. Published 2021 Jul 14. doi: 10.1021/acs.jmedchem.1c00480.

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88

Unknown

Mechanisms of the Antiproliferative and Antitumor Activity of Novel Telomerase–Carbonic Anhydrase Dual-Hybrid Inhibitors (2021)

Plyasova, Anna A. ; Berrino, Emanuela ; Khan, Irina I. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11432-11444. Published 2021 Jul 20. doi: 10.1021/acs.jmedchem.1c00756.

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89

Unknown

Issue Publication Information (2021)

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): jmv064i015_1503723. Published 2021 Aug 12. doi: 10.1021/jmv064i015_1503723.

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90

Unknown

Discovery of TAK-041: a Potent and Selective GPR139 Agonist Explored for the Treatment of Negative Symptoms Associated with Schizophrenia (2021)

Reichard, Holly A. ; Schiffer, Hans H. ; Monenschein, Holger ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11527-11542. Published 2021 Jul 14. doi: 10.1021/acs.jmedchem.1c00820.

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91

Unknown

Structural Insights into Notum Covalent Inhibition (2021)

Zhao, Yuguang ; Svensson, Fredrik ; Steadman, David ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11354-11363. Published 2021 Jul 22. doi: 10.1021/acs.jmedchem.1c00701.

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Publication Date: 2021-07-22

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92

Unknown

Design, Synthesis, and Biological Evaluation of Organic Nitrite (NO2–) Donors as Potential Anticerebral Ischemia Agents (2021)

Wu, Jianbing ; Yin, Wei ; Huang, Zhangjian ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 10919-10933. Published 2021 Jul 22. doi: 10.1021/acs.jmedchem.1c00282.

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93

Unknown

Recent Progress and Clinical Development of Inhibitors that Block MDM4/p53 Protein–Protein Interactions (2021)

Zhang, Shiyan ; Lou, Jianfeng ; Li, Yafang ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 10621-10640. Published 2021 Jul 21. doi: 10.1021/acs.jmedchem.1c00940.

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94

Unknown

Gut-Restricted Selective Cyclooxygenase-2 (COX-2) Inhibitors for Chemoprevention of Colorectal Cancer (2021)

Zhang, Zhuming ; Ghosh, Avijit ; Connolly, Peter J. ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11570-11596. Published 2021 Jul 19. doi: 10.1021/acs.jmedchem.1c00890.

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95

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Structure-Based Optimization of ML300-Derived, Noncovalent Inhibitors Targeting the Severe Acute Respiratory Syndrome Coronavirus 3CL Protease (SARS-CoV-2 3CLpro) (2021)

Han, Sang Hoon ; Goins, Christopher M. ; Arya, Tarun ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; acs.jmedchem.1c00598. Published 2021 Aug 04. doi: 10.1021/acs.jmedchem.1c00598. [early online release]

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96

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Discovery of the First Selective M4 Muscarinic Acetylcholine Receptor Antagonists with in Vivo Antiparkinsonian and Antidystonic Efficacy (2021)

Moehle, Mark S. ; Bender, Aaron M. ; Dickerson, Jonathan W. ; [et al.]

American Chemical Society

In: ACS Pharmacology . 2021; 4(4): 1306-1321. Published 2021 Aug 02. doi: 10.1021/acsptsci.0c00162.

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97

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Design, Optimization, and Structural Characterization of an Apoptosis-Inducing Factor Peptide Targeting Human Cyclophilin A to Inhibit Apoptosis Inducing Factor-Mediated Cell Death (2021)

Russo, Luigi ; Mascanzoni, Fabiola ; Farina, Biancamaria ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11445-11459. Published 2021 Aug 02. doi: 10.1021/acs.jmedchem.1c00777.

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98

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Xanthine Derivatives Reveal an Allosteric Binding Site in Methylenetetrahydrofolate Dehydrogenase 2 (MTHFD2) (2021)

Lee, Lung-Chun ; Peng, Yi-Hui ; Chang, Hsin-Huei ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11288-11301. Published 2021 Aug 02. doi: 10.1021/acs.jmedchem.1c00663.

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99

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Announcing the Latest Inductees to the ACS Division of Medicinal Chemistry Hall of Fame (2021)

Schwarz, Jacob B.

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 10517-10518. Published 2021 Aug 03. doi: 10.1021/acs.jmedchem.1c01288.

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100

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Are Pt(IV) Prodrugs That Release Combretastatin A4 True Multi-action Prodrugs? (2021)

Schmidt, Claudia ; Babu, Tomer ; Kostrhunova, Hana ; [et al.]

American Chemical Society

In: Journal of Medicinal Chemistry. 2021; 64(15): 11364-11378. Published 2021 Aug 03. doi: 10.1021/acs.jmedchem.1c00706.

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