ExLibris header image
SFX Logo
Title: Identification and optimisation of a series of substituted 5-pyridin-2-yl-thiophene-2-hydroxamic acids as potent histone deacetylase (HDAC) inhibitors
Source:

Bioorganic & Medicinal Chemistry Letters [0960-894X] Price, Steve yr:2007


Collapse list of basic services Basic
Sorry, no full text available...
Please use the document delivery service (see below)  
Holding information
Holdings in library search engine ALBERT GO
Document delivery
Request document via Library/Bibliothek GO
Users interested in this article also expressed an interest in the following:
1. HAYAKAWA, M. "Synthesis and biological evaluation of 4-morpholino-2-phenylquinazolines and related derivatives as novel PI3 kinase p110α inhibitors." Bioorganic & medicinal chemistry 14.20 (2006): 6847-5844. Link to SFX for this item
2. Sun, D. "Synthesis and optimization of novel 4,4-disubstituted cyclohexylbenzamide derivatives as potent 11 beta-HSD1 inhibitors." Bioorganic and medicinal chemistry letters 21.1 (2011): 405-410. Link to SFX for this item
3. Drogemuller, M. "Synthesis of cephalostatin analogues by symmetrical and non-symmetrical routes." European journal of organic chemistry 12 (1998): 2811-2831. Link to Full Text for this item Link to SFX for this item
4. Suzuki, T. "Non-hydroxamate histone deacetylase inhibitors." Current medicinal chemistry 12.24 (2005): 2867-2880. Link to SFX for this item
5. Bauser, M. "Discovery and optimization of 2-aryl oxazolopyrimidines as adenosine kinase inhibitors using liquid phase parallel synthesis." Bioorganic & medicinal chemistry letters 14.8 (2004): 1997-2000. Link to SFX for this item
6. Pretzer, D. "Stability of the experimental anticancer agent [[(4-methoxyphenyl)sulfonyl]hydrazono]acetic acid (NSC-267213). II. Effect of structural modification on stability and mechanism of degradation." International Journal of Pharmaceutics 38.1 (1987): 161-169. Link to Full Text for this item Link to SFX for this item
7. Zheng, X. "Analgesic agents without gastric damage: Design and synthesis of structurally simple benzenesulfonanilide-type cyclooxygenase-1-selective inhibitors." Bioorganic & medicinal chemistry 15.2 (2007): 1014-1021. Link to SFX for this item
8. Gauuan, Polivina a. "Superoxide dismutase mimetics: synthesis and structure-activity relationship study of MnTBAP analogues." Bioorganic & medicinal chemistry 10.9 (2002): 3013-21. Link to Full Text for this item Link to SFX for this item
9. Suzuki, T. "Rational design of non-hydroxamate histone deacetylase inhibitors." Mini reviews in medicinal chemistry 6.5 (2006): 515-526. Link to SFX for this item
10. Chapman, M. n. "Optimizing the pharmacology of statins: characteristics of rosuvastatin." Atherosclerosis. Supplements 2.4 (2002): 33-37. Link to SFX for this item
11. KNIGHT, Zachary A. "Isoform-specific phosphoinositide 3-kinase inhibitors from an arylmorpholine scaffold." Bioorganic & medicinal chemistry 12.17 (2004): 4749-59. Link to SFX for this item
12. Guo, W. "Synthesis and biological assays of 9-(acylamino) homocamptothecins as DNA topoisomerase I inhibitors." Chemistry & biodiversity 10.10 (2013): 1804-15. Link to Full Text for this item Link to SFX for this item
13. Flessner, T. "N,N′-Bis(3,5-di-t-butylsalicylidene)-1,2-cyclohexanediamino-manganese(III) chloride - the Jacobsen catalyst." Journal für praktische Chemie 341.5 (1999): 436-444. Link to Full Text for this item Link to SFX for this item
14. Axten, J. "Discovery of 7-Methyl-5-(1-{[3-(trifluoromethyl)phenyl]acetyl}-2,3-dihydro-1H-indol-5-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine (GSK2606414), a Potent and Selective First-in-Class Inhibitor of Protein Kinase R (PKR)-like Endoplasmic Reticulum Kinase (PERK)." Journal of medicinal chemistry 55.16 (2012): 7193-7207. Link to Full Text for this item Link to SFX for this item
15. Reardon, David A. "Phase I study of AEE788, a novel multitarget inhibitor of ErbB- and VEGF-receptor-family tyrosine kinases, in recurrent glioblastoma patients." Cancer chemotherapy and pharmacology 69.6 (2012): 1507-1518. Link to Full Text for this item Link to SFX for this item
16. Funabashi, K. "Enantioselective construction of quaternary stereocenter through a reissert-type reaction catalyzed by an electronically tuned bifunctional catalyst: Efficient synthesis of various biologically significant compounds." Journal of the American Chemical Society 123.43 (2001): 10784-10785. Link to Full Text for this item Link to SFX for this item
17. Martin-Kohler, A. "Furo[2,3-d]pyrimidines and oxazolo[5,4-d]pyrimidines as inhibitors of receptor tyrosine kinases (RTK)." Helvetica chimica acta 87.4 (2004): 956-975. Link to Full Text for this item Link to SFX for this item
18. Wetzel, M. "Effect of trichostatin A, a histone deacetylase inhibitor, on glioma proliferation in vitro by inducing cell cycle arrest and apoptosis." Journal of neurosurgery 103.6 (2006): 549-56. Link to SFX for this item
19. Mander, Lewis N. "Total Synthesis of Sordaricin." Journal of organic chemistry 70.5 (2005): 1654-1670. Link to Full Text for this item Link to SFX for this item
20. Miller, Thomas A. "Histone deacetylase inhibitors." Journal of medicinal chemistry 46.24 (2003): 5097-5116. Link to Full Text for this item Link to SFX for this item
View More...
View Less...
Select All Clear All

Expand list of advanced services Advanced