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Synthesis of 1,5-benzodiazepine heterocycles containing a trifluoromethyl group

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Chemistry of Heterocyclic Compounds Aims and scope

Summary

2,3-Dihydro-1,5-benzodiazepines containing a trifluoromethyl group were obtained by the reaction of α,β-unsaturated ketones CF3COCH=CR1R2 with o-phenylenediamine.

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Authors
  1. V. G. Nenajdenko
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  2. A. V. Sanin
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  3. E. S. Balenkova
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Additional information

M. V. Lomonosov State University, Moscow 119899. Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 10. pp. 1429–1431, October, 1994. Original article October 11, 1994.

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Nenajdenko, V.G., Sanin, A.V. & Balenkova, E.S. Synthesis of 1,5-benzodiazepine heterocycles containing a trifluoromethyl group. Chem Heterocycl Compd 30, 1240–1242 (1994). https://doi.org/10.1007/BF01184893

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  • DOI: https://doi.org/10.1007/BF01184893

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