Publication Date:
2005-01-18
Description:
〈br /〉〈span class="detail_caption"〉Notes: 〈/span〉Cole, Stewart T -- Alzari, Pedro M -- New York, N.Y. -- Science. 2005 Jan 14;307(5707):214-5.〈br /〉〈span class="detail_caption"〉Author address: 〈/span〉Genetique Moleculaire Bacterienne and Biochimie Structurale Units, Institut Pasteur, Paris 75724 Cedex 15, France. stcole@pasteur.fr〈br /〉〈span class="detail_caption"〉Record origin:〈/span〉 〈a href="http://www.ncbi.nlm.nih.gov/pubmed/15653490" target="_blank"〉PubMed〈/a〉
Keywords:
Adenosine Triphosphate/biosynthesis
;
Animals
;
Antitubercular Agents/chemistry/*pharmacology/therapeutic use
;
Bacterial Proton-Translocating ATPases/*antagonists &
;
inhibitors/chemistry/metabolism
;
Clinical Trials, Phase II as Topic
;
Diarylquinolines
;
Drug Design
;
Drug Evaluation, Preclinical
;
Drug Resistance, Bacterial
;
Enzyme Inhibitors/pharmacology/therapeutic use
;
Humans
;
Mice
;
Microbial Sensitivity Tests
;
Mycobacterium smegmatis/drug effects/genetics
;
Mycobacterium tuberculosis/*drug effects/enzymology/genetics
;
Protein Structure, Secondary
;
Proton-Motive Force
;
Proton-Translocating ATPases/chemistry/metabolism
;
Quinolines/chemistry/*pharmacology/therapeutic use
;
Tuberculosis/*drug therapy/microbiology
;
Tuberculosis, Multidrug-Resistant/*drug therapy/microbiology
Print ISSN:
0036-8075
Electronic ISSN:
1095-9203
Topics:
Biology
,
Chemistry and Pharmacology
,
Computer Science
,
Medicine
,
Natural Sciences in General
,
Physics
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