ExLibris header image
SFX Logo
Title: Structure-based design of novel groups for use in the P1 position of thrombin inhibitor scaffolds. Part 1: Weakly basic azoles
Source:

Bioorganic & Medicinal Chemistry Letters [0960-894X] Isaacs, Richard C.A. yr:2006


Collapse list of basic services Basic
Sorry, no full text available...
Please use the document delivery service (see below)  
Holding information
Holdings in library search engine ALBERT GO
Document delivery
Request document via Library/Bibliothek GO
Users interested in this article also expressed an interest in the following:
1. Wagner, J. "Rational Design, Synthesis, and X-ray Structure of Selective Noncovalent Thrombin Inhibitors." Journal of medicinal chemistry 41.19 (1998): 3664-3674. Link to Full Text for this item Link to SFX for this item
2. Medina, J. "Optimization of a series of quinazolinone-derived antagonists of CXCR3." Bioorganic & medicinal chemistry letters 19.17 (2009): 5114-5118. Link to SFX for this item
3. Muley, L. "Think Twice: Understanding the High Potency of Bis(phenyl)methane Inhibitors of Thrombin." Journal of molecular biology 391.3 (2009): 552-564. Link to SFX for this item
4. Neochoritis, C. "1-Arylaminoimidazole-2-thiones as Intermediates in the Synthesis of Imidazo[2,1-b][1,3,4]thiadiazines." Tetrahedron 64.16 (2008): 3527-. Link to SFX for this item
5. BEKKALI, Y. "Identification of a novel class of succinyl-nitrile-based Cathepsin S inhibitors." Bioorganic & medicinal chemistry letters 17.9 (2007): 2465-2749. Link to SFX for this item
6. Noeske-Jungblut, C. "Triabin, a highly potent exosite inhibitor of thrombin." The Journal of biological chemistry 270.48 (1995): 28629-28634. Link to SFX for this item
7. Muley, L. "Enhancement of hydrophobic interactions and hydrogen bond strength by cooperativity: Synthesis, modeling, and molecular dynamics simulations of a congeneric series of thrombin inhibitors." Journal of medicinal chemistry 53.5 (2010): 2126-2135. Link to Full Text for this item Link to SFX for this item
8. Hattori, K. "Rational design of conformationally restricted quinazolinone inhibitors of poly(ADP-ribose)polymerase." Bioorganic & medicinal chemistry letters 17.20 (2007): 5577-5581. Link to SFX for this item
9. CALVINOCASILDA, V. "Sonocatalysis and zeolites: An efficient route to prepare N-alkylimidazoles." Applied catalysis 338.1 (2008): 130-135. Link to SFX for this item
10. Yan, Z. "A close inspection of Ag(I) coordination to molecular baskets. A study of solvation and guest encapsulation in solution and the solid state." Tetrahedron 65.35 (2009): 7213-7219. Link to SFX for this item
11. Casas-Solvas, L. "Ferrocene-beta-Cyclodextrin Conjugates: Synthesis, Supramolecular Behavior, and Use as Electrochemical Sensors." Chemistry : a European journal 15.33 (2009): 8146-8162. Link to Full Text for this item Link to SFX for this item
12. Al-Obaid, A. "Substituted quinazolines, part 3. Synthesis, in vitro antitumor activity and molecular modeling study of certain 2-thieno-4(3H)-quinazolinone analogs." European Journal of Medicinal Chemistry 44.6 (2009): 2379-2391. Link to SFX for this item
13. Lee, Yeon n. "Understanding the structural requirements of 4-anilidopiperidine analogues for biological activities at μ and δ opioid receptors." Bioorganic & medicinal chemistry letters 17.8 (2007): 2161-2165. Link to SFX for this item
14. Johnson, M. "Discovery and optimization of a series of quinazolinone-derived antagonists of CXCR3." Bioorganic & medicinal chemistry letters 17.12 (2007): 3339-3343. Link to SFX for this item
15. KOCHANNY, Monica J. "Substituted thiophene-anthranilamides as potent inhibitors of human factor Xa." Bioorganic & medicinal chemistry 15.5 (2007): 2127-2146. Link to SFX for this item
16. del Rio, Fu-Yao E. "Highly enantioselective oxidation of sulfides to sulfoxides by a new oxaziridinium salt." Organic letters 9.12 (2007): 2265-2268. Link to Full Text for this item Link to SFX for this item
17. Srisiri, W. "Influence of Lewis Acids on the Cycloaddition Reactions of Cyano- and Carbomethoxy-Substituted Olefins." Journal of organic chemistry 59.18 (1994): 5424-5435. Link to Full Text for this item Link to SFX for this item
18. Luppi, G. "A new entry to polyfunctionalized 4,5-trans disubstituted oxazolidin-2-ones from L-aspartic acid." Synlett 2003.6 (2003): 797-800. Link to SFX for this item
19. Westerlund, A. "Investigation of 1-bromo-3-buten-2-one as building block in organic synthesis." Tetrahedron 57.27 (2001): 5879-5883. Link to Full Text for this item Link to SFX for this item
20. IWAKUBO, M. "Design and synthesis of rho kinase inhibitors (III)." Bioorganic & medicinal chemistry 15.2 (2007): 1022-1033. Link to SFX for this item
View More...
View Less...
Select All Clear All

Expand list of advanced services Advanced
A service provided by the Library of the Wissenschaftspark Albert Einstein, Potsdam, Germany.
© 2005 SFX by Ex Libris Inc.